II. Interactions: Metabolized by CYP1A2 (Substrates)

III. Interactions: Inhibitor of CYP1A2

  1. Neuropsychiatric Drugs
    1. Fluvoxamine (Luvox)
    2. Tacrine (Cognex)
  2. Cardiopulmonary Drugs
    1. Verapamil
    2. Diltiazem
    3. Amiodarone (inhibitor)
  3. Antibiotics
    1. Enoxacin: Inhibitor
    2. Ciprofloxacin: Inhibitor
    3. Norfloxacin: Inhibitor
  4. Miscellaneous Drugs
    1. Grapefruit juice
    2. Cimetidine
    3. Ticlopidine

IV. Interactions: Inducers of CYP1A2

  1. Neuropsychiatric drugs
    1. Phenobarbital
    2. Phenytoin
  2. Antibiotics
    1. Rifampin
  3. Miscellaneous
    1. Charcoal broiled beef
    2. Tobacco exposure (e.g. Cigarette smoke)
    3. Cruciferous vegetables
    4. Omeprazole (Prilosec)

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