Human Immunodeficiency Virus Book

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Fusion Inhibitor

Aka: Fusion Inhibitor, Enfuvirtide, Fuzeon
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  1. See Also
    1. Anti-Retroviral Therapy
  2. Class
    1. Anti-retroviral agent
    2. Fusion Inhibitor
  3. Indications
    1. Treatment-experienced patients
    2. Limited use in clinical practice
  4. Mechanism
    1. Blocks HIV to chemokine receptor binding on CD4 cells
  5. Adverse Effects
    1. Injection site pain and reaction (common)
    2. Eosinophilic Hypersensitivity Reaction (<1%)
    3. Neutropenia
    4. Increased risk of Bacterial Pneumonia
  6. References
    1. (2009) Treat Guidel Med Lett 7(78): 11-22
    2. Reust (2011) Am Fam Physician 83(12): 1443-51

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