II. Indications
- Replaced by Second Generation Sulfonylurea agents for the management of Type II Diabetes Mellitus
III. Preparations
- Acetohexamide (Dymelor)
- Dose: 500-750 mg qd or divided ($14)
- Chlorpropamide (Diabinese)
- Dose: 100-250 up to 750 mg qd/bid
- Antidiuretic effect (used in Diabetes Insipidus)
- Tolazamide (Tolinase)
- Dose: 250-500 mg PO qd or divided ($2.81)
- Tolbutamide (Orinase)
- Dose: 1000-2000mg qd or divided bid ($2.75)